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GRIN1

GRIN1 NMDA receptor — the molecular target that 1 compounds in the wiki act on.

In one line: A learning-and-memory receptor that ketamine blocks — with a rapid antidepressant effect.

GRIN1 is part of the NMDA receptor, central to learning and memory. Ketamine blocks it, which paradoxically triggers a surge of brain growth signals (BDNF) and rapidly regrows lost connections — lifting severe depression within hours instead of the weeks antidepressants take.

That's why a form of ketamine is now an approved treatment for depression that hasn't responded to other drugs. It's given under supervision because blocking this receptor also causes a dissociative, dream-like state.

Compounds acting on GRIN1