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Cromoglicic acid

  • Prescription medicine
  • Prescription only
  • Identity checked
  • Sources last checked 2026-09-04

This page shows what was measured, who it was measured in, and what that does not settle.

What Cromoglicic acid does in the body

Most allergy drugs block the receiver of the histamine signal.

This one was designed to stop the signal being sent: to make the cells that store histamine less willing to release it when they meet an allergen. Because it barely gets absorbed, it only works on whatever surface you apply it to — the nose, the eye, the airway lining — and it has to be there before the allergen arrives. Exactly how it calms those cells has never been settled.

Why people take it. Preventing asthma attacks, hay fever and itchy eyes before they start — and, by mouth, the gut symptoms of mastocytosis

What happened in people

No statistically significant difference from placebo on percentage of symptom-free days across four pooled paediatric asthma trials

Source-linked record

Where this came from

A person wrote this into the record with the study named beside it. No reviewer has signed it off.

The recorded finding that sits closest to something a person would notice. Written into the record, not signed off, and it carries no population or interval.

The limit that matters most

Only six products remain in the CMS acquisition survey, the smallest count of any drug in this batch, at $0.5845 per millilitre

Where it acts
The mucosal surface it is applied to — bronchial epithelium, nasal mucosa, conjunctiva, or gut lumen. Almost none of it is absorbed, which is the whole design
Kind of result
Symptoms and quality of life
Supervision
RNAWiki has not recorded a supervision or regulatory status for this substance.

What the registries record it as

  • The substance registry classes this as chemical.

    FDA substance registry · Y0TK0FS77W · read 2026-08-29

  • Its recorded molecular formula is C23H14Na2O11, weighing 512.34.

    US prescribing information · 00623958-a8fe-47d1-a0d2-0aa4e2f7966e · read 2026-08-30

Where each sentence above came from

A person wrote this explanation into the record, with the studies named in the path below.

The recorded use, written for a reader without medical training. Not signed off.

A limit recorded against this substance. Not signed off as a reviewed claim.

The four opening statements run to 115 words.

Words this page uses

Four words worth knowing first

Chosen from what this page shows, with each one explained before the word it depends on.

Placebo

A placebo is a dummy treatment given so the real one can be compared with it.

A picture of it, and where the picture fails

A placebo is like a blank control in an experiment.

Where that stops being true. A blank does nothing. People given a placebo often do get better.

What people get wrong. A placebo effect is read as imaginary. The improvement is measured and real.

An inactive intervention matched in appearance to the test intervention, used to control for non-specific effects.

Comparator

A comparator is whatever the treatment was measured against.

A picture of it, and where the picture fails

It is like the other runner in a race.

Where that stops being true. A race has one winner. A study can show both arms improved.

What people get wrong. Results are read without asking what the other group got. Beating nothing is not beating a treatment.

The control condition against which the experimental intervention is assessed.

Randomisation

Randomisation means chance decides who gets which treatment.

A picture of it, and where the picture fails

It is like a coin toss deciding the groups.

Where that stops being true. A coin toss is fair once. Fairness here comes from doing it for everyone.

What people get wrong. It is thought to make groups identical. It makes them similar on average, including on things nobody measured.

Allocation of participants to arms by a chance process, so that unmeasured factors are balanced in expectation.

What happened in peopleRead from sources, not yet reviewed

What happened in people

Each card is one study: the exact question it asked, who was in it, and whether it showed what it set out to show.

Efficacy of sodium cromoglycate against placebo as maintenance therapy in children aged 0 to 18

The study did not show it

Who was studied
Cochrane CD002173.pub2 — inhaled sodium cromoglycate for asthma in children
How many people
1026
Study design
Systematic review and meta-analysis of 23 double-blind placebo-controlled trials
Compared against
A dummy treatment
Kind of result
A number that stands in for health
What was found
No statistically significant difference on percentage of symptom-free days; other symptom outcomes significant with small effects; funnel plot indicating publication bias
Repeated elsewhere
Failed to Replicate

What this does not prove. A study that did not show an effect does not show that no effect exists anywhere.

The limits of this study, and where it came from

Main limit. Trials published 1970 to 1997, mostly crossover, few reporting allocation concealment. The authors state publication bias is likely to have overestimated the beneficial effects.

How far it carries. This study is recorded from the curated record, not from the registry match.

Form and route. Four route-specific formulations: inhalation solution for nebulisation, nasal solution over the counter, ophthalmic solution, and oral concentrate

Interval reported. Not recorded in this summary

Written into the record, not signed off as a reviewed claim.

Participant-reported severity of ocular itching, irritation, tearing and photophobia

The study showed what it set out to show

Who was studied
Cochrane CD009566.pub2 — topical antihistamines and mast cell stabilisers
How many people
4344
Study design
Systematic review of 30 randomised trials across 17 drugs or comparisons
Compared against
Not recorded for this study
Kind of result
A number that stands in for health
What was found
All reported agents, cromoglicate among them, reduced symptoms and signs against placebo in the short term; no serious adverse events reported for the class
Repeated elsewhere
Partially Replicated

What this does not prove. Meeting one endpoint in one population does not carry to other goals or other people.

The limits of this study, and where it came from

Main limit. Treatment periods of one to eight weeks only, with no long-term efficacy data for any drug in the class. Meta-analysis was possible for one comparison, which did not involve cromoglicate.

How far it carries. This study is recorded from the curated record, not from the registry match.

Form and route. Four route-specific formulations: inhalation solution for nebulisation, nasal solution over the counter, ophthalmic solution, and oral concentrate

Interval reported. Not recorded in this summary

Written into the record, not signed off as a reviewed claim.

What we know
RNAWiki holds 2 written-up human studies for this substance, each with the question it asked.
How we know it
Each card names the study, the number of people and what the study set out to measure.
What this does not prove
These summaries were written by a person and have not been signed off as reviewed claims.
Why it matters
A study that failed is as informative as one that worked, and both are here.
What we still do not know
No reviewed claim exists, so no exact population, effect size or interval is published yet.

What it changes in the bodyRead from sources, not yet reviewed

The path through the body

From what a person takes to what changes. A solid line is a step measured in people. A dashed line is a step nobody has measured that way.

  1. Start

    Cromoglicic acid

    What a person takes: Four route-specific formulations: inhalation solution for nebulisation, nasal solution over the counter, ophthalmic solution, and oral concentrate.

    The measurement behind this step

    Each formulation treats only the surface it reaches, because the molecule is not absorbed. All require dosing several times daily to maintain local concentration, since there is no plasma half-life doing that work. The inhalation label describes it as a prophylactic given on a regular daily basis, with effect usually evident after several weeks though some patients respond almost immediately.

  2. Getting in

    Applied to a surface, and it stays there

    Sprayed into the nose, nebulised into the lungs, dropped into the eye, or swallowed to reach the gut lining. Which formulation you use decides which surface is treated, because none of it travels.

    Described, with no measurement named. No measurement is named for this step, so it is drawn as an unconfirmed link.

    The measurement behind this step

    Two carboxylic acids fully ionised at physiological pH give a doubly anionic molecule with negligible absorption across any epithelium. Four separate route-specific formulations exist for that reason, and the oral concentrate acts on gut mucosal mast cells without entering the circulation.

  3. Reaching the cell

    It never enters the cell

    The molecule is far too charged to cross a cell membrane. Whatever it does, it does from the outside — which is one reason the mechanism has been so hard to pin down.

    Described, with no measurement named. No measurement is named for this step, so it is drawn as an unconfirmed link.

    The measurement behind this step

    The double negative charge that prevents systemic absorption equally prevents passive entry into mast cells. Any mechanism must therefore operate at the cell surface or through a surface receptor, which is what makes the GPR35 hypothesis structurally attractive and the classical membrane-stabilisation account structurally awkward.

  4. What it acts on

    The classical account: the mast cell is stabilised

    The traditional explanation is that it makes the mast cell membrane less likely to open and release its contents when an allergen arrives. This is the phrase the whole drug category is named after.

    Described, with no measurement named. No measurement is named for this step, so it is drawn as an unconfirmed link.

    The measurement behind this step

    Early studies attributed the cromones’ prevention of allergic reactions to mast cell stabilising properties. The 2017 review states the exact pharmacological mechanism remained a mystery, and that the account cannot explain the discrepancies between species and between mast cell subtypes in their response to the drugs.

  5. The change it makes

    Two candidate mechanisms, neither settled

    One idea is that the drug activates a specific receptor on the cell surface. The other is that it boosts one of the body’s own anti-inflammatory systems, the one steroids also use. Both have evidence and neither has closed the question.

    Measured in animals. A result in animals says what to test next. It does not say what happens in people.

    The measurement behind this step

    Cromoglycate, nedocromil and zaprinast increase inositol phosphate accumulation and calcium mobilisation in HEK cells transfected with the orphan receptor GPR35, though its relevance to mast cell mediator release is unelucidated. Separately, cromones potentiate glucocorticoid-induced annexin A1 release by inhibiting PP2A phosphatase, and annexin A1 depletion in vitro completely reverses their inhibitory actions.

  6. What that does for a person

    The allergic reaction is smaller, if it is prevented in advance

    Used regularly and started before exposure, less histamine is released and the reaction is milder. Used during a reaction it does nothing, because it works upstream of everything that is already happening.

    Measured in people. Written by a person from the study named beside the step. Not signed off as a reviewed claim.

    The measurement behind this step

    The inhalation label describes it as a prophylactic agent given on a regular daily basis, with effect usually evident after several weeks though some patients respond almost immediately. There is no receptor-blocking component, so nothing in the mechanism addresses mediators already released.

  7. What that does for a person

    What the pooled trials actually showed

    On the cleanest measure in childhood asthma — days with no symptoms — pooling the trials found no difference from placebo, and the shape of the published literature suggested negative studies were missing.

    Described, with no measurement named. No measurement is named for this step, so it is drawn as an unconfirmed link.

    The measurement behind this step

    Twenty-three trials in 1,026 children published 1970 to 1997; percentage of symptom-free days showed no statistically significant difference; other symptom outcomes reached significance with small effects and wide intervals; funnel plot indicated under-representation of small negative studies.

No suggested links are held for this record, so nothing is hidden from this path.

What we know
The record describes 6 steps from taking it to an effect in a person.
How we know it
Each step names the study behind it in the technical detail beside it.
What this does not prove
A change inside the body is a reason to look. It is not a result in a person.
Why it matters
A reader can see exactly where the chain stops being measured in people.
What we still do not know
No reviewed claim binds any of these steps to a named population.

What is missing or unclearRead from sources, not yet reviewed

Were people like you studied?

RNAWiki cannot tell whether a study fits you. It can show who was in it, and where the result stops carrying.

Who was studied

People similar to this profile were included.

  • Historically children with asthma, and still people with allergic rhinitis and allergic conjunctivitis over the counter. The oral concentrate is used for mastocytosis, where the target cell is unambiguously the mast cell.

Who is missing from the studies

  • Which groups were under-represented in the studies has not been recorded for this substance. Pregnancy, breastfeeding, children, older adults, and people with liver or kidney conditions are commonly excluded from trials; nothing here says whether they were.

What the label states about particular groups

  • On pediatric, the label states: “In adult rats no adverse effects of cromolyn sodium were observed at oral doses up to 6144 mg/kg (approximately 25 times the maximum recommended daily oral dose in adults on a mg/m 2 basis).”

    US prescribing information · 00623958-a8fe-47d1-a0d2-0aa4e2f7966e · read 2026-08-30

  • On older people, the label states: “Clinical studies of GASTROCROM did not include sufficient numbers of subjects aged 65 and over to determine whether they respond differently from younger subjects.”

    US prescribing information · 00623958-a8fe-47d1-a0d2-0aa4e2f7966e · read 2026-08-30

  • On people who are pregnant, the label states: “There are, however, no adequate and well controlled studies in pregnant women.”

    US prescribing information · 00623958-a8fe-47d1-a0d2-0aa4e2f7966e · read 2026-08-30

  • On people who are breastfeeding, the label states: “It is not known whether this drug is excreted in human milk.”

    US prescribing information · 00623958-a8fe-47d1-a0d2-0aa4e2f7966e · read 2026-08-30

Where the result stopped carrying

  • The pooled percentage of symptom-free days in childhood asthma showed no significant difference from placebo
  • Publication bias was detected in the paediatric asthma literature, with small negative studies under-represented
  • The drug lost its place as maintenance therapy for childhood asthma from 1990 onward as inhaled corticosteroids arrived
  • Every original brand — Intal, Opticrom, Crolom — has left the active Drugs@FDA product listing
  • This is a scope explorer, not a diagnosis engine.
  • It shows who was studied so you can see whether people similar to you were included.

RNAWiki cannot tell whether a study fits you. It can show who was in it.

What it would be like to takeRead from sources, not yet reviewed

Why it might seem to do nothing

A real effect and a noticed effect are different things. These are the recorded reasons the two come apart.

It was studied in different people

The people in the studies were not much like the reader.

On this record: Which groups were under-represented in the studies has not been recorded for this substance. Pregnancy, breastfeeding, children, older adults, and people with liver or kidney conditions are commonly excluded from trials; nothing here says whether they were.

The evidence may simply be wrong

Small early studies often do not hold up.

On this record: RNAWiki has not yet published a reviewed conclusion for this use.

Other reasons RNAWiki checked and found nothing for (11)
It was studied for a different goal
The studies measured something else entirely. Nothing in this record points to this reason.
A different form was studied
The studied form is not the form on the shelf. Nothing in this record points to this reason.
There was nothing to correct
Where a level is already normal, topping it up may change nothing. Nothing in this record points to this reason.
Something else had to happen too
In the studies it was paired with training, a diet or another treatment. Nothing in this record points to this reason.
The change is too small to feel
A real change can still sit below what a person notices. Nothing in this record points to this reason.
Day-to-day swing hides it
Sleep, food, stress and time of day move most numbers more than this would. Nothing in this record points to this reason.
Not enough time yet
The studies ran longer than the person has waited. Nothing in this record points to this reason.
It was not taken as studied
Missed days change the result, and studies count them. Nothing in this record points to this reason.
Something else changed at the same time
Two changes at once cannot be told apart afterwards. Nothing in this record points to this reason.
The product may not be what it says
Contents of a sold product are not always what the label states. Nothing in this record points to this reason.
No recorded reason
RNAWiki has nothing stored that would explain it. Nothing in this record points to this reason.

None of these is a reason to take more. Taking more is not a step this page ever suggests.

What it would be like to takeRead from sources, not yet reviewed

What taking it involves

The recorded facts about getting hold of it and using it. Nothing here is a suggestion about what you should do.

How it is supplied

Prescription only

Quoted from a source

Where this came from

Copied from a source RNAWiki stored, with the source named.

Read from the recorded approval status.

No source is stored against this line.

Form and route

Four route-specific formulations: inhalation solution for nebulisation, nasal solution over the counter, ophthalmic solution, and oral concentrate

Source-linked record

Where this came from

A person wrote this into the record with the study named beside it. No reviewer has signed it off.

The form and route recorded on this substance.

No source is stored against this line.

Who oversees it

RNAWiki has not recorded a supervision or regulatory status for this substance.

Quoted from a source

Where this came from

Copied from a source RNAWiki stored, with the source named.

No register row and no identity class settled the question.

No source is stored against this line.

What is in the pack

Each formulation treats only the surface it reaches, because the molecule is not absorbed. All require dosing several times daily to maintain local concentration, since there is no plasma half-life doing that work. The inhalation label describes it as a prophylactic given on a regular daily basis, with effect usually evident after several weeks though some patients respond almost immediately.

Source-linked record

Where this came from

A person wrote this into the record with the study named beside it. No reviewer has signed it off.

Recorded notes on how this is sold and what that means for what is in the pack.

No source is stored against this line.

Where it is registered

Regulatory records are listed in the technical disclosure at the foot of this page.

Counted from records

Where this came from

A count of rows RNAWiki holds. It describes our records, not your body.

Register entries are stored per jurisdiction and shown with their dates.

No source is stored against this line.

Why people stop

Not recorded.

Nothing recorded

Where this came from

RNAWiki holds nothing here and says so rather than guessing.

No record of why people stopped taking it is stored for this substance.

No source is stored against this line.

What it would be like to takeRead from sources, not yet reviewed

What can go wrong

Sorted by where each line came from. A regulator's label and a report somebody sent in are not the same kind of fact.

Worth asking a clinician aboutWritten into the record from the studies named on this page

Among the most benign safety profiles in this batch, and for a structural reason: a doubly anionic molecule that is essentially not absorbed cannot produce systemic toxicity. The Cochrane review of topical antihistamines and mast cell stabilisers reported no serious adverse events related to the class across 30 trials in 4,344 participants. Local irritation on application — throat irritation and cough with inhalation, nasal stinging and sneezing with the spray, transient burning with the drops — is the practical limit. The safety record is the strongest thing about this drug and it was never the reason it was displaced.

Nobody counted how many people took this and were fine, so this cannot be turned into a rate.

Where this came from

Over a long time. No completed tested study window is recorded, so long-term effects are not established by the registry record.

Groups the studies covered thinly. Which groups were under-represented in the studies has not been recorded for this substance. Pregnancy, breastfeeding, children, older adults, and people with liver or kidney conditions are commonly excluded from trials; nothing here says whether they were.

What is missing or unclearRead from sources, not yet reviewed

Does the exact form matter?

Evidence belongs to the exact thing that was tested. A different salt, a different mixture or a different preparation is a different question.

The form that was studied

Four route-specific formulations: inhalation solution for nebulisation, nasal solution over the counter, ophthalmic solution, and oral concentrate

Source-linked record

Where this came from

A person wrote this into the record with the study named beside it. No reviewer has signed it off.

The form used in the studies cited on this page.

No source is stored against this line.

What is sold

All require dosing several times daily to maintain local concentration, since there is no plasma half-life doing that work. The inhalation label describes it as a prophylactic given on a regular daily basis, with effect usually evident after several weeks though some patients respond almost immediately.

Source-linked record

Where this came from

A person wrote this into the record with the study named beside it. No reviewer has signed it off.

Recorded notes on which forms are sold and how they compare.

No source is stored against this line.

What is recorded as being sold

  • 27 products list this as an active ingredient in the United States drug directory. 27 of them contain it and nothing else.

    FDA National Drug Code directory · 42571-445 · read 2026-08-29

  • They are sold as liquid, powder, solution, solution, concentrate, solution/ drops and spray, metered, taken intrabronchial, nasal, ophthalmic and oral.

    FDA National Drug Code directory · 42571-445 · read 2026-08-29

  • The regulator's established pharmacologic class for it is decreased histamine release [pe] and mast cell stabilizer [epc].

    FDA National Drug Code directory · 42571-445 · read 2026-08-29

  • 11 published labels name it as an active ingredient. 11 of them describe this substance alone, which is where its own label text on this page comes from.

    US prescribing information · 93f80edb-3b38-423e-8cd6-5b5cb4393ec2 · read 2026-08-29

  • Those labels are classed as human otc drug and human prescription drug.

    US prescribing information · 93f80edb-3b38-423e-8cd6-5b5cb4393ec2 · read 2026-08-29

  • Gastrocrom is oral at HOW SUPPLIED GASTROCROM Oral Concentrate is an unpreserved, colorless solution supplied in a low density polyethylene plastic unit dose ampule with 8 ampules per foil pouch., recorded as fda label in effect 2024-06-26 in the United States.

    US prescribing information · 00623958-a8fe-47d1-a0d2-0aa4e2f7966e · read 2026-08-30

  • Recorded price in US: 0.33569–0.98098 USD per one millilitre, across 8 priced products whose strengths and pack forms differ, as of 2026-08-26, paid by retail pharmacies buying the product, as surveyed by the Centers for Medicare & Medicaid Services. It is not a list price, an insurance price, or what anyone pays at a counter..

    Recorded source · 2026-08-26 · read 2026-08-28

Evidence carries across two names for one substance. It does not carry across a salt, a mirror form or a mixture.

What it would be like to takeRead from sources, not yet reviewed

What you could measure

This one is decided with a clinician, so this section holds questions to ask rather than a plan to run.

RNAWiki could not confidently classify this substance, so no self-experiment plan is offered.

Questions worth asking

  • Which of the trials of Cromoglicic acid studied people like me?
  • What was measured, and for how long?
  • Was the result a laboratory value or a health outcome?
  • What would we watch for, and when would we stop?

Tracking can show whether something changed for you. It cannot show what caused it.

RNAWiki records evidence. It does not say whether this substance is right for you.

What is missing or unclearRead from sources, not yet reviewed

Claims that go past the evidence

Things said about this substance that sound reasonable, and the exact step that is missing between the evidence and the claim.

Goes past the evidence

That "mast cell stabiliser" describes a known mechanism — the 2017 review calls the exact mechanism a mystery and notes species and subtype discrepancies the account cannot explain

Why it sounds right. It follows from something real on this page: a body step, an animal result or a related finding.

The missing step. Nobody measured this in people for this use, or the study that did measure it did not show it.

What would change this

A study in people, for this exact use, measuring this exact thing, that a reviewer signs off.

RNAWiki has not yet published a reviewed conclusion for this use.

Goes past the evidence

That the statistically significant secondary symptom outcomes in childhood asthma reflect a real effect, given the publication bias the funnel plot indicates

Why it sounds right. It follows from something real on this page: a body step, an animal result or a related finding.

The missing step. Nobody measured this in people for this use, or the study that did measure it did not show it.

What would change this

A study in people, for this exact use, measuring this exact thing, that a reviewer signs off.

RNAWiki has not yet published a reviewed conclusion for this use.

Goes past the evidence

That the GPR35 findings translate into therapeutic effect — the review states explicitly that it is unclear how they would

Why it sounds right. It follows from something real on this page: a body step, an animal result or a related finding.

The missing step. Nobody measured this in people for this use, or the study that did measure it did not show it.

What would change this

A study in people, for this exact use, measuring this exact thing, that a reviewer signs off.

RNAWiki has not yet published a reviewed conclusion for this use.

Goes past the evidence

That a mast-cell rationale established in mastocytosis transfers to asthma, where the pooled primary outcome was null

Why it sounds right. It follows from something real on this page: a body step, an animal result or a related finding.

The missing step. Nobody measured this in people for this use, or the study that did measure it did not show it.

What would change this

A study in people, for this exact use, measuring this exact thing, that a reviewer signs off.

RNAWiki has not yet published a reviewed conclusion for this use.

What is missing or unclearRead from sources, not yet reviewed

What nobody knows yet

Open questions, each with why it is open and what would close it.

Missing populations

Which groups were under-represented in the studies has not been recorded.

Why it matters. Recorded by the evidence model as a gap on this record.

What would answer it

A study that measures it, and a reviewer to sign it off.

Last checked 2026-09-04. Searched: The sources listed in the receipts at the foot of this page.

Missing long-term data

No completed tested study window is recorded.

Why it matters. Recorded by the evidence model as a gap on this record.

What would answer it

A study that measures it, and a reviewer to sign it off.

Last checked 2026-09-04. Searched: The sources listed in the receipts at the foot of this page.

No reviewed conclusion

RNAWiki has not yet published a reviewed conclusion for this use.

Why it matters. Recorded by the evidence model as a gap on this record.

What would answer it

A study that measures it, and a reviewer to sign it off.

Last checked 2026-09-04. Searched: The sources listed in the receipts at the foot of this page.

Missing interaction studies

No interaction was found in the registers checked. Not finding one is not the same as showing there is none.

Why it matters. Recorded by the evidence model as a gap on this record.

What would answer it

A study that measures it, and a reviewer to sign it off.

Last checked 2026-09-04. Searched: The sources listed in the receipts at the foot of this page.

Formulation uncertainty

Several salts, forms or products of Cromoglicic acid are recorded. Results from one form may not transfer to another.

Why it matters. Recorded by the evidence model as a gap on this record.

What would answer it

A study that measures it, and a reviewer to sign it off.

Last checked 2026-09-04. Searched: The sources listed in the receipts at the foot of this page.

Mechanism not reviewed

No reviewed mechanism story exists for this substance.

Why it matters. Recorded by the evidence model as a gap on this record.

What would answer it

A study that measures it, and a reviewer to sign it off.

Last checked 2026-09-04. Searched: The sources listed in the receipts at the foot of this page.

What happened in peopleRead from sources, not yet reviewed

Check any of this yourself

Every line above traced back to the study it came from. This is the technical layer, and the vocabulary changes here.

Every line above can be traced to the study named beside it. Follow the link and read it.

Cochrane: no significant benefit on symptom-free days, and the missing studies were the negative ones
In plain words
Twenty-three trials in a thousand children were pooled. On the cleanest measure — how many days a child had no symptoms — the drug was no better than placebo. The pattern of published studies showed that small trials with negative results were missing from the literature.
What was measured
Percentage of symptom-free days, pooled across four trials, cromoglycate against placebo
Effect estimate
No reviewed effect estimate exists for this record.
Limits
This entry records a failure.
From the source
The Cochrane review searched for all double-blind placebo-controlled randomised trials of inhaled sodium cromoglycate as maintenance therapy in children aged 0 to 18 with asthma, screening 3,500 titles and including 24 papers reporting 23 studies published between 1970 and 1997, together enrolling 1,026 participants. Most were crossover studies and few provided enough information to judge allocation concealment. Four studies reported percentage of symptom-free days; pooling them revealed no statistically significant difference between cromoglycate and placebo. Other pooled symptom outcomes and bronchodilator use reached statistical significance but with small treatment effects, and the confidence intervals were wide enough that a clinically relevant effect could not be excluded either. The funnel plot showed an under-representation of small studies with negative results, indicating publication bias. The authors concluded there is insufficient evidence to be sure about efficacy over placebo, and that publication bias is likely to have overestimated the beneficial effects.
Source
van der Wouden JC, Uijen JH, Bernsen RM, Tasche MJ, de Jongste JC, Ducharme F. Cochrane Database Syst Rev 2008;4:CD002173
Role in the trial
Not matched to a registered study
Identity check
no open identity hold
Audit mark
verified
Review state
Written into the record, not signed off as a reviewed claim
The mechanism that named a whole drug class has never been established
In plain words
Cromolyn is the original "mast cell stabiliser" and the phrase was invented for it. Nearly sixty years after it was made, the pharmacologists reviewing it wrote that the exact mechanism remained a mystery.
What was measured
That cromolyn works by stabilising the mast cell membrane — the phrase that defines the class, offered without a confirmed molecular mechanism and contradicted by species and subtype discrepancies its own reviewers describe
Effect estimate
No reviewed effect estimate exists for this record.
Limits
See the technical detail.
From the source
A 2017 review by researchers including one of the original pharmacologists in the field states that while early studies attributed the cromones’ ability to prevent allergic reactions to their mast cell stabilising properties, the exact pharmacological mechanism by which this occurred remained a mystery, and that the classical account cannot explain the discrepancies between species and between mast cell subtypes in their response to these drugs. Two candidate mechanisms are advanced. First, the orphan G-protein coupled receptor GPR35: cromoglycate, nedocromil and zaprinast increase inositol phosphate accumulation and calcium mobilisation in HEK cells transfected with GPR35, though the review notes its significance to asthma, allergy or mast cell mediator release is yet to be elucidated and it is unclear how those actions would translate into therapeutic effect. Second, the annexin A1 and formyl peptide receptor anti-inflammatory loop: cromones potentiate glucocorticoid-induced annexin A1 release by inhibiting PP2A phosphatase activity, and depletion of annexin A1 in vitro completely reverses their inhibitory actions.
Source
Sinniah A, Yazid S, Flower RJ. Front Pharmacol 2017;8:827
Role in the trial
Not matched to a registered study
Identity check
no open identity hold
Audit mark
contested
Review state
Written into the record, not signed off as a reviewed claim
It was displaced from asthma by a class with better evidence, not by a safety finding
In plain words
This drug was standard maintenance treatment for childhood asthma for years. Its use fell away from 1990 as inhaled steroids took over. Nothing dangerous was discovered — the replacement simply had evidence that held up.
What was measured
That a drug leaving practice implies it was found harmful — here it was displaced by a comparator with stronger evidence while remaining one of the safest molecules in respiratory medicine
Effect estimate
No reviewed effect estimate exists for this record.
Limits
See the technical detail.
From the source
The Cochrane review records that sodium cromoglycate was recommended as maintenance treatment for childhood asthma for many years and that its use decreased after 1990 when inhaled corticosteroids became popular, while still being used in many countries. The displacement was not driven by any safety signal: cromolyn remains among the best-tolerated drugs in respiratory medicine, and the Cochrane review of topical antihistamines and mast cell stabilisers in allergic conjunctivitis, which included cromoglicate, reported no serious adverse events for the class. What changed was the availability of a comparator whose evidence base did not depend on trials published between 1970 and 1997 with a funnel plot showing missing negatives. Every original brand — Intal, Opticrom, Crolom — has since left the active Drugs@FDA product listing.
Source
van der Wouden JC et al., Cochrane Database Syst Rev 2008;4:CD002173, Background; Drugs@FDA product listings for cromolyn sodium
Role in the trial
Not matched to a registered study
Identity check
no open identity hold
Audit mark
verified
Review state
Written into the record, not signed off as a reviewed claim
It is essentially not absorbed, and that is the design
In plain words
The molecule carries two permanent negative charges, so almost none of it crosses from the gut or the airway into the bloodstream. It can only act on the surface you put it on — which is why there are four different formulations for four different surfaces.
What was measured
Ionisation state and route-specific formulation set, from structure and regulatory listings
Effect estimate
No reviewed effect estimate exists for this record.
Limits
See the technical detail.
From the source
Cromoglicic acid is a symmetrical bis-chromone with two carboxylic acid groups, fully ionised at physiological pH, giving a doubly anionic molecule with negligible passive membrane permeability. The consequence runs through the whole product family: separate formulations exist for inhalation, nasal, ophthalmic and oral routes, and the oral concentrate is indicated for mastocytosis precisely because it acts on gut mucosal mast cells without being absorbed. It also explains the safety record — a drug that does not enter the circulation cannot produce systemic toxicity — and the dosing burden, since local concentration must be maintained by repeated application rather than by a plasma half-life.
Source
PubChem CID 2882, structure and physicochemical properties; Drugs@FDA route listings for cromolyn sodium (inhalation, nasal, ophthalmic, oral)
Role in the trial
Not matched to a registered study
Identity check
no open identity hold
Audit mark
verified
Review state
Written into the record, not signed off as a reviewed claim
Across the eye-drop class it works, in the short term, like everything else
In plain words
In allergic conjunctivitis, the systematic review that examined every drop in this class found that all of them beat a dummy in the short term, including this one, and that none of them has any long-term data.
What was measured
Participant-reported ocular symptom severity against placebo, class-wide across 30 trials
Effect estimate
No reviewed effect estimate exists for this record.
Limits
See the technical detail.
From the source
The Cochrane review of topical antihistamines and mast cell stabilisers for seasonal and perennial allergic conjunctivitis identified 30 randomised trials in 4,344 participants across 17 drugs or comparisons, with nedocromil sodium and sodium cromoglycate among the agents evaluated. Overall risk of bias was low but reporting quality variable and outcome reporting highly heterogeneous; meta-analysis was possible for only one comparison, which did not involve cromoglicate. The conclusion was that all reported agents reduce symptoms and signs of seasonal allergic conjunctivitis against placebo in the short term, that trials evaluated treatment periods of one to eight weeks only with no long-term efficacy data, and that no serious adverse events related to the class were reported.
Source
Castillo M, Scott NW, Mustafa MZ, Mustafa MS, Azuara-Blanco A. Cochrane Database Syst Rev 2015;6:CD009566
Role in the trial
Not matched to a registered study
Identity check
no open identity hold
Audit mark
verified
Review state
Written into the record, not signed off as a reviewed claim
The one indication where the target cell is beyond doubt is the smallest one
In plain words
For mastocytosis — a disease defined by too many mast cells — the oral form has its own approval. That is the only place where "mast cell drug" is not an assumption about the mechanism but a description of the disease.
What was measured
That a mast-cell-directed rationale transfers from mastocytosis, where the cell type defines the disease, to asthma, where the Cochrane review found no significant effect on symptom-free days
Effect estimate
No reviewed effect estimate exists for this record.
Limits
See the technical detail.
From the source
Gastrocrom, cromolyn sodium oral concentrate, was approved under NDA 020479 on 29 February 1996 and remains the only branded cromolyn product in the active Drugs@FDA listing, with generics from 2011 onward. In mastocytosis the pathology is an excess of mast cells, so the drug and the disease are matched at the level of the cell type regardless of which molecular mechanism turns out to be correct — the therapeutic rationale does not depend on resolving the GPR35 or annexin A1 question. This is a narrower and firmer claim than the one made for the inhaled product, where the same cell type is one participant among many in a complex inflammatory disease.
Source
Drugs@FDA: GASTROCROM (cromolyn sodium) oral concentrate, NDA 020479, approved 29 February 1996
Role in the trial
Not matched to a registered study
Identity check
no open identity hold
Audit mark
caution
Review state
Written into the record, not signed off as a reviewed claim

Where else this substance is registered

FDA substance identifier (UNII)
Y0TK0FS77W
CAS registry number
16110-51-3
PubChem compound
2882
ChEMBL
CHEMBL428880
ChEBI
59039
WHO international nonproprietary name list entry
2427
RxNorm concept
42612
EMA substance identifier
100000083740
European Chemicals Agency number
240-279-8
DrugBank
DB01003

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    Trial roles classified for highlighted evidence

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    Safety mode resolved

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    Canonical metadata present

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What is missing or unclearRead from sources, not yet reviewed

How this medicine reached us

Kept near the foot of the page. A historical event moves up only when it changes something about this substance today.

What the approval register records

  • 31 approved applications cover products containing this substance. The earliest was NDA018596, approved 19820528 to KING PHARMS LLC.

    Drugs@FDA application register · NDA018596 · read 2026-08-29

  • Marketing status on the register: discontinued, over-the-counter and prescription.

    Drugs@FDA application register · NDA018596 · read 2026-08-29

  • The earliest marketing start date recorded for a listed product is 19930217.

    FDA National Drug Code directory · 42571-445 · read 2026-08-29

What is missing or unclearRead from sources, not yet reviewed

What to learn next

Ordered by what would most change how you read this page, starting with what is easiest to misunderstand.

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What is not here

7 questions this page could not answer

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  • Felt, measured, or meaningful — found nothing in the sources checked.
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The record as stored

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Everything above is built from what is below. This layer keeps the technical vocabulary, record identifiers and every stored row, so a reader who wants to check the page can.

The older medicine-wide conclusion held in this record

Written for a clinical reader, and about the medicine as a whole rather than about one indication, population and set of trials. RNAWiki does not treat it as a programme conclusion and no reviewer has signed it off in that form. It is here word for word because it is what the record holds.

A bis-chromone so poorly absorbed that it only works where it is sprayed — the drug that named the mast cell stabiliser class, whose mechanism its own pharmacologists called a mystery as recently as 2017, and whose Cochrane review of 23 trials in 1,026 children found no significant difference from placebo on symptom-free days with a funnel plot showing missing small negative studies.

Recorded evidence blocks (9)

On the Cromoglicic acid label: indicated for what?


"GASTROCROM is indicated in the management of patients with mastocytosis. Use of this product has been associated with improvement in diarrhea, flushing, headaches, vomiting, urticaria, abdominal pain, nausea, and itching in some patients.": indications and usage on Cromoglicic acid's label. DailyMed label · 00623958-a8fe-47d1-a0d2-0aa4e2f7966e · 2024-06-26

23 registered trials of Cromoglicic acid — at which phases?


Registered studies posting no result
20 of 23

23 registered studies of Cromoglicic acid: 10 phase2, 5 phase1, 4 phase3, 2 early phase1, 2 phase4, 1 na, 1 na or unstated. CLINICALTRIALS_SNAPSHOT · 2026-09-01

254 with a PubMed record

Show the evidence
  • phase2
    10
  • phase1
    5
  • phase3
    4
  • early phase1
    2
  • phase4
    2
  • na
    1
8 more recorded rows
  • na or unstated
    1
  • completed
    8
  • terminated
    6
  • not yet recruiting
    3
  • recruiting
    3
  • enrolling by invitation
    1
  • unknown
    1
  • withdrawn
    1

recorded 2026-09-01 · last checked 2026-09-04

7 of Cromoglicic acid's trials stopped: futility/efficacy, accrual/recruitment, other?


futility/efficacy (1), accrual/recruitment (4) and other (2): Cromoglicic acid's stop wording, clustered. CLINICALTRIALS_SNAPSHOT · 2026-09-01

"prematurely terminated because of low recruitment"; 7 of 23 registered studies

Show the evidence

Trial

  • NCT01701843
    terminated; "prematurely terminated because of low recruitment"
  • NCT01841307
    terminated; "Difficulty recruiting; Funding ended; interim analysis provided sufficient data for interpretation."
  • NCT02664051
    terminated; "Inactive"
  • NCT03202147
    withdrawn; "Study halted prematurely prior to initiation but potentially will resume in the future."
  • NCT04408664
    terminated; "Insufficient accrual rate"
  • NCT04428775
    terminated; "Low enrollment"
  • 1 further recorded trial NCT05077917
    terminated; "slow enrollment"

recorded 2026-09-01 · last checked 2026-09-04

Human studies of Cromoglicic acid used Cromolyn Sodium (17.1 mg BID) — over how long?


Human studies of Cromoglicic acid used "Cromolyn Sodium (17.1 mg BID)". ClinicalTrials.gov · 2026-09-01

Show the evidence
  • human NCT07142291
    Cromolyn Sodium (17.1 mg BID)

recorded 2026-09-01 · last checked 2026-09-04

Which running trial of Cromoglicic acid could settle function?


NCT07757555 measures Change in Physical Function as Measured by the PROMIS® Physical Function Scale, reading out 2028-02-02.

1 open trial; n 25; "Guanfacine and Cromolyn Sodium for POTS: The DBPOTS Trial"

Show the evidence
  • Trial NCT07757555
    "Guanfacine and Cromolyn Sodium for POTS: The DBPOTS Trial"; n 25; "Change in Physical Function as Measured by the PROMIS® Physical Function Scale"; 2028-02-02

Which 5 trials of Cromoglicic acid posted no result?


Posted no result
5 of 5 completed trials
Registrations
NCT00745199, NCT01722812, NCT02566252, NCT02547818 and NCT03167216
Completion dates
oldest 2009-06; newest 2022-06-30
Show the evidence

Trial

  • NCT00745199
    2009-06
  • NCT01722812
    2013-05
  • NCT02566252
    2016-03
  • NCT02547818
    2020-11-18
  • NCT03167216
    2022-06-30

At the median, Cromoglicic acid's trials enrolled 21 people — anything larger?


Median enrolment
21
Largest enrolment
5000
Registered trials counted
22

What do 8 spontaneous reports say about Cromoglicic acid — and not say?


These are reports people sent to a regulator. They do not show the medicine caused the reaction. Nobody counted how many people took the medicine and reported nothing. The same event can be reported more than once, and many reports are incomplete. News coverage, lawsuits and new warnings change how often people report. A count is not a rate and not a risk.

Cromoglicic acid appears in spontaneous reports to regulators. Across the 1 most-reported reaction term, 8 reaction mentions were counted: treatment failure 8. FAERS via Open Targets · CHEMBL428880 · 2026-06-24

Show the evidence
  • treatment failure
    8

recorded 2026-06-24 · last checked 2026-09-04

Which reaction does Cromoglicic acid's label not list?


treatment failure reported for Cromoglicic acid, absent from its label. FAERS via Open Targets · CHEMBL428880 · 2026-06-24

2 label terms; 1 reported and unlisted; 00623958-a8fe-47d1-a0d2-0aa4e2f7966e

Show the evidence
  • treatment failure
    count not stated

recorded 2026-06-24 · last checked 2026-09-04

Where it is registered
Identifiers, relations and other names

The exact record

ChEMBL id
CHEMBL428880
PubChem CID
2882
CAS number
16110-51-3
RxCUI
42612
InChIKey
IMZMKUWMOSJXDT-UHFFFAOYSA-N
Also called
CROMOLYN, Acide cromoglicique, Acido cromoglicico, Cromo-comod, Cromoglicate, Cromoglycate, alzt-op1a, CROMOLYN SODIUM, Astilyn, Natrii cromoglicas, rvt-1601
Development code
R03BC01, FPL-670, NSC-109500
Trade name
Aerocrom, Allercrom, Aspire, Brol-eze, Catacrom, Clariteyes, Crolom, Cromogen, Cromogen e-breathe, Cromolux, Cromoptic, Cromosol
Salt form
Cromoglicate sodium, Cromolyn disodium salt, Disodium cromolyn, Sodium cromoglicate, Sodium cromoglycate, Sodium cromolyn
British name
Cromoglycic acid
Sources (6)

Sources

ChEMBL 37 — CC BY-SA 3.0 Unported · ChEMBL ATC CC BY-SA · ClinicalTrials.gov — US Government work · Open Targets 26.06 — CC0 · mixed register set; per-register licences in docs/specs/corpus-20k-sources.md · openFDA / DailyMed — US Government work

How these records are assembled · Which registers were checked

Index-quality checks
  • identity passed: no open identity hold
  • required summary fields resolved: 4 required field(s) not terminal: Why people use it, Best-supported result, Biggest unanswered question, Human evidence
  • public claims reviewed: 0 reviewed claim(s); drafts are never rendered
  • source coverage passed: 6 source rows
  • no critical contamination: no quarantine open
  • canonical metadata passed: slug and display name present
  • no raw internal fields: enforced by the copy-contract test over the rendered page

This is a record of evidence. It is not medical advice, and it does not say this substance suits you. Nothing here says any substance on RNAWiki is appropriate for a child.